Ingredients Anti-aging Caffeine
49Cf
Tier · Moderate evidence
Anti-aging · Antioxidant

Caffeine

INCI: Caffeine · Also called: 1,3,7-Trimethylxanthine

Tightens and brightens the under-eye area, reducing the look of puffiness by constricting tiny blood vessels. Best deployed in eye creams.

For your skin

Tightens and brightens the under-eye area, reducing the look of puffiness by constricting tiny blood vessels. Best deployed in eye creams.

Want the science? Keep reading ↓

Mechanism of action

Methylxanthine that vasoconstricts capillaries, inhibits phosphodiesterase to stimulate lipolysis, and scavenges free radicals.

Why we tier this moderate

6 cited papers across 3 countries. The mechanism is well-described and there's at least one controlled trial in the literature, but we tier this Moderate rather than Strong to stay honest about how many specific papers we cite directly.

4
International
1
European Union
1
Korea

Cited research

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Elias M et al., Caffeine in Skincare: Its Role in Skin Cancer, Sun Protection, and Cosmetics, Indian Journal of Dermatology 2023;68(5):546-550 — evidence for topical caffeine's photoprotective, antioxidant, and anti-cellulite roles

2023Meta-analysis — positivePMID:38099120View source ↗
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Gherardini J et al. (Germany), Transepidermal UV radiation of scalp skin ex vivo induces hair follicle damage that is alleviated by the topical treatment with caffeine, International Journal of Cosmetic Science 2019;41(2):164-182 — topical caffeine reduced UV-induced hair follicle cytotoxicity and premature catagen entry in ex vivo human scalp

2019Positive — efficacyPMID:30746733View source ↗
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Byun SY et al., Efficacy of Slimming Cream Containing 3.5% Water-Soluble Caffeine and Xanthenes for the Treatment of Cellulite, Annals of Dermatology 2015;27(3):243-249 — 3.5% caffeine slimming cream improved visual cellulite scores 19.8% with measurable circumference reductions over 6 weeks

2015Positive — efficacyPMID:26082579View source ↗
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Luo L, Lane ME (UK), Topical and transdermal delivery of caffeine, International Journal of Pharmaceutics 2015;490(1-2):155-64 — review of caffeine physicochemistry and formulation strategies for skin permeation supporting cosmetic and transdermal use

2015Mechanism onlyPMID:26004004View source ↗
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Herman A, Herman AP, Caffeine's mechanisms of action and its cosmetic use, Skin Pharmacology and Physiology 2013;26(1):8-14 — vasoconstriction, antioxidant, lipolysis; 3% topical caffeine penetrates skin barrier effectively

2013Mechanism onlyPMID:23075568View source ↗
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Lupi O et al., Evaluation of the effects of caffeine in the microcirculation and edema on thighs and buttocks using orthogonal polarization spectral imaging and clinical parameters, Journal of Cosmetic Dermatology 2007;6(2):102-107 — 7% topical caffeine significantly reduced thigh/hip circumference

2007Positive — efficacyPMID:17524126View source ↗

Sources: PubMed · KCI · J-Stage · CNKI · Wanfang · SFD · MFDS · Cochrane · SCCS · CIR. Every entry points to a specific document. See methodology for what each outcome label means.